Papers - TAKAO Koichi
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Syntheses and evaluation of 2- or 3-(N-cyclicamino)chromone derivatives as monoamine oxidase inhibitors Reviewed
Koichi Takao, Tsukasa Sakatsume, Hitoshi Kamauchi and Yoshiaki Sugita
Chem.Pharm.Bull. 68 ( 11 ) 1082 - 1089 2020.11
Authorship:Lead author Language:English Publishing type:Research paper (scientific journal) Publisher:Bulletins of the Pharmaceutical Society of Japan
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Synthesis and pharmacological evaluation of childinin E and several derivatives as anti-hyphal formation inhibitors against Candida albicans. Reviewed International journal
Hitoshi Kamauchi Momoka Hirata, Koichi Takao, Yoshiaki Sugita
Tetrahedron Letters 61 ( 49 ) 152588 2020.10
Language:English Publishing type:Research paper (scientific journal)
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Quantification of the ability of natural products to prevent herpes virus infection Reviewed International journal
Kunihiko Fukuchi, Hiroshi Sakagami, Yoshiaki Sugita, Koichi Takao, Daisuke Asai, Shigemi Terakubo, Hiromu Takemura, Hirokazu Ohno, Misaki Horiuchi, Madoka Suguro, Tomohiro Fujisawa, Kazuki Toeda, Hiroshi Oizumi, Toshikazu Yasui, Takaaki Oizumi
Medicines 7 ( 64 ) 2020.10
Language:English Publishing type:Research paper (scientific journal) Publisher:MDPI
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Syntheses and crystal structures of two piperine derivatives. Reviewed International journal
Toshinari Ezawa, Yutaka Inoue, Isamu Murata, Mitsuaki Suzuki, Koichi Takao, Yoshiaki Sugita, Ikuo Kanamoto
Acta Crystallogr. E. Crystallogr. Commun. 76 ( 5 ) 646 - 650 2020.05
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of 2-Arylazolylchromones and 2-Triazolylchromones. Reviewed
Junko Nagai, Haixia Shi, Natsuko Sezaki, Nao Yoshida, Kenjiro Bandow, Yoshihiro Uesawa, Hiroshi Sakagami, Mineko Tomomura, Akito Tomomura, Koichi Takao, Yoshiaki Sugita
Anticancer Res. 2019.12
Language:English Publishing type:Research paper (scientific journal)
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Further Quantitative Structure–Cytotoxicity Relationship Analysis of 3-Styrylchromones Reviewed
Koichi Takao, Kaori Hoshi, Hiroshi Sakagami, Haixia Shi, Kenjiro Bandow, Junko Nagai, Yoshihiro Uesawa, Akito Tomomura, Mineko Tomomura, Yoshiaki Sugita
Anticancer Res. 2019.12
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of 2-Styrylchromones Reviewed
Yoshihiro Uesawa, Junko Nagai, Haixiaa Shi, Hiroshi Sakagami, Kenjiro Bandow, Akito Tomomura, Mineko Tomomura, Saki Endo, Koichi Takao, Yoshiaki Sugita
Anticancer Res. 2019.12
Language:English Publishing type:Research paper (scientific journal)
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2-Styrylchromone derivatives as potent and selective monoamine oxidase B inhibitors. Reviewed
Koichi Takao, Saki Endo, Junko Nagai, Hitoshi Kamauchi, Yuri Takemura, Yoshihiro Uesawa, Yoshiaki Sugita
Bioorganic Chemistry 2019.11
Authorship:Lead author Language:English Publishing type:Research paper (scientific journal)
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Synthesis of natural product-like polyprenylated phenols and quinones: evaluation of their neuroprotective activities. Reviewed
Hitoshi Kamauchi, Takumi Oda, Kanayo Horiuchi, Koichi Takao, Yoshiaki Sugita
Bioorganic Medicinal Chemistry 2019.11
Language:English Publishing type:Research paper (scientific journal)
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Design, synthesis and evaluation of 2-(indolylmethylidene)-2,3-dihydro-1-benzofuran-3-one and 2-(indolyl)-4H-chromen-4-one derivatives as novel monoamine oxidases inhibitors. Reviewed
Koichi Takao, Shiori U, Hitoshi Kamauchi, Yoshiaki Sugita
Bioorganic Chemistry 2019.06
Authorship:Lead author Language:English Publishing type:Research paper (scientific journal)
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Synthesis and biological evaluation of pyrano[4,3-b][1]benzopyranone derivatives as monoamine oxidase and cholinesterase inhibitors. Reviewed
Koichi Takao, Yuka Kubota, Hitoshi Kamauchi and Yoshiaki Sugita
Bioorganic Chemistry 2019.03
Authorship:Lead author Language:English Publishing type:Research paper (scientific journal)
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Extracellular spermine activates DNA methyltransferase 3A and 3B. Reviewed
Taro Fukui, Kuniyasu Soda, Koichi Takao, Toshiki Rikiyama
Int. J. Mol. Sci. 2019.03
Language:English Publishing type:Research paper (scientific journal)
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Evaluation of the molecular state of piperine in cyclodextrin complexes by near-infrared spectroscopy and solid-state fluorescence measurements Reviewed International journal
Toshinari Ezawa, Yutaka Inoue, Isamu Murata, Koichi Takao, Yoshiaki Sugita, Ikuo Kanamoto
International Journal of Medicinal Chemistry 2019.02
Language:English Publishing type:Research paper (scientific journal) Publisher:Hindawi
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Protective Effects of Brain Infarction by N-Acetylcysteine Derivatives Reviewed
Takeshi Uemura, Kenta Watanabe, Kyohei Higashi, Noriyuki Kogure, Mariko Kitajima, Hiromitsu Takayama, Koichi Takao, Yoshiaki Sugita, Akihiko Sakamoto, Yusuke Terui, Toshihiko Toida, Keiko Kashiwagi, and Kazuei Igarashi
Stroke 49 ( 7 ) 1727 - 1733 2018.07
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of 2-(N-cyclicamino)chromone derivatives Reviewed
Haixia Shi, Junko Nagai, Tsukasa Sakatsume, Kenjiro Bandow, Noriyuki Okudaira, Hiroshi Sakagami, Mineko Tomomura, Akito Tomomura, Yoshihiro Uesawa, Koichi Takao and Yoshiaki Sugita
Anticancer Res. 38 ( 7 ) 3897 - 3906 2018.07
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of Furo[2,3-b]chromones Reviewed
Yoshihiro Uesawa, Hiroshi Sakagami, Haixia Shi, Maria Hirose, Koichi Takao and Yoshiaki Sugita
Anticancer Res. 38 ( 6 ) 3283 - 3290 2018.06
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of Pyrano[4,3-b]chromones Reviewed
Junko Nagai, Haixia Shi, Yuka Kubota, Kenjiro Bandow, Noriyuki Okudaira, Yoshihiro Uesawa, Hiroshi Sakagami, Mineko Tomomura, Akito Tomomura, Koichi Takao and Yoshiaki Sugita
Anticancer Res. 2018
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of 3-(N-Cyclicamino)chromone Derivatives Reviewed
Haixia Shi, Junko Nagai, Tsukasa Sakatsume, Kenjiro Bandow, Noriyuki Okudaira, Yoshihiro Uesawa, Hiroshi Sakagami, Mineko Tomomura, Akito Tomomura, Koichi Takao and Yoshiaki Sugita
Anticancer Res. 2018
Language:English Publishing type:Research paper (scientific journal)
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Characterization of the dissolution behavior of piperine/cyclodextrins inclusion complexes Reviewed
Ezawa T, Inoue Y, Murata I, Takao K, Sugita Y, Kanamoto I
AAPS Pharm. Sci. Tech. 2018
Language:English Publishing type:Research paper (scientific journal)
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Quantitative Structure–Cytotoxicity Relationship of 2-Azolylchromones Reviewed
Hiroshi Sakagami, Noriyuki Okudaira, Yoshihiro Uesawa, Koichi Takao, Hajime Kagaya, Yoshiaki Sugita
Anticancer Res. 2018
Language:English Publishing type:Research paper (scientific journal)