Papers - TAKAO Koichi
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Caldomycin, a new guanidopolyamine produced by a novel agmatine homocoupling enzyme involved in homospermidine biosynthesis. Reviewed International coauthorship
Teruyuki Kobayashi, Akihiko Sakamoto, Tamao Hisano, Keiko Kashiwagi, Kazuei Igarashi, Koichi Takao, Takeshi Uemura, Takemitsu Furuchi, Yoshiaki Sugita, Toshiyuki Moriya, Tairo Oshima and Yusuke Terui
Sci. Rep. 14 ( 1 ) 7566 2024.03
Language:English Publishing type:Research paper (scientific journal)
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Synthesis of 2,8-Dioxabicyclo[3.3.1]nonane Derivatives and Their Neuroprotective Activities Reviewed
Hitoshi Kamauch, Akifumi Takanashi, Mitsuaki Suzuki, Kouki Izumi, Koichi Takao, Yoshiaki Sugita
Chem.Pharm.Bull. 72 ( 1 ) 56 - 60 2024.01
Language:English Publishing type:Research paper (scientific journal) Publisher:Bulletins of the Pharmaceutical Society of Japan
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Synthesis and biological evaluation of 2-azolylmethylene-3-(2H)-benzofuranone derivatives as potent monoamine oxidases inhibitors Reviewed
Koichi Takao, Yuka Kubota, Kota Kurosaki, Hitoshi Kamauchi, Yoshihiro Uesawa, Yoshiaki Sugita
Chem.Pharm.Bull. 72 ( 1 ) 109 - 120 2024.01
Authorship:Lead author, Corresponding author Language:English Publishing type:Research paper (scientific journal) Publisher:Bulletins of the Pharmaceutical Society of Japan
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A Tricyclic Aromatic Polyketide Isolated from the Marine-derived Fungus Curvularia aeria Reviewed
Hitoshi Kamauchi, Mayu Tanaka, Mitsuaki Suzuki, Miho Furukawa, Atsushi Ikeda, Chihiro Sasho, Yuka Kiba, Masashi Kitamura, Koichi Takao, Yoshiaki Sugita
Chem.Pharm.Bull. 72 ( 1 ) 98 - 101 2024.01
Language:English Publishing type:Research paper (scientific journal) Publisher:Bulletins of the Pharmaceutical Society of Japan
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Intracellular polyamine depletion induces N-linked galactosylation of the monoclonal antibody produced by CHO DP-12 cells. Reviewed
Rin Miyajima, Hitomi Manaka, Tatsuya Honda, Noritaka Hashii, Masato Suzuki, Masahiro Komeno, Koichi Takao, Akiko Ishii-Watabe, Kazuei Igarashi, Toshihiko Toida, Kyohei Higashi
J. Biotechnol. 378 1 - 10 2023.11
Language:English Publishing type:Research paper (scientific journal) Publisher:Bulletins of the Pharmaceutical Society of Japan
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Inclusion complexes of Ursolic acid with Cyclodextrin-based metal-organic Framework-1 enhance its solubility. Reviewed International coauthorship
Yutaka Inoue, Ayana Motoda, Takashi Tanikawa, Koichi Takao, Florencio Arce Jr., Gerard Lee See, Yoshiyuki Ishida, Daisuke Nakata, Keiji Terao
Journal of Drug Delivery Science and Technology 89 104986 2023.10
Language:English Publishing type:Research paper (scientific journal)
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Inhibition of Polyamine Catabolism Reduces Cellular Senescence Reviewed
Takeshi Uemura, Miki Matsunaga, Yuka Yokota, Koichi Takao, Takemitsu Furuchi
Int. J. Mol. Sci. 24 ( 17 ) 13397 2023.08
Language:English Publishing type:Research paper (scientific journal)
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Potentiation of Anticancer Activity of G2/M Blockers by Mild Hyperthermia Reviewed
Yuya Tagawa, Hiroshi Sakagami, Sei-Ichi Tanuma, Shigeru Amano, Shin Uota, Kenjiro Bandow, Mineko Tomomura, Yoshihiro Uesawa, Koichi Takao, Yoshiaki Sugita, Nobuharu Yamamoto, Hideaki Sakashita, Rina Nakakaji, Toshiyuki Koizumi, Kenji Mitsudo, Iwai Tohnai
Anticancer Res. 43 ( 8 ) 3429 - 3439 2023.08
Language:English Publishing type:Research paper (scientific journal)
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Putrescine Biosynthesis from Agmatine by Arginase (TtARG) in Thermus thermophilus Reviewed International journal
Teruyuki Kobayashi, Akihiko Sakamoto, Keiko Kashiwagi, Kazuei Igarashi, Koichi Takao, Takeshi Uemura, Toshiyuki Moriya, Tairo Oshima, Yusuke Terui
J. Biochem. 2023.07
Language:English Publishing type:Research paper (scientific journal) Publisher:Oxford University Press
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A Comparative Study of Tumor-specificity and Neurotoxicity between 3-Styrylchromones and Anticancer Drugs Reviewed
Tomoyuki Abe, Hiroshi Sakagami, Shigeru Amano, Shin Uota, Kenjiro Bandow, Yoshihiro Uesawa, Shiori U, Hiroki Shibata, Yuri Takemura, Yu Kimura, Koichi Takao, Yoshiaki Sugita, Akira Sato, Sei-Ichi Tanuma, Hiroshi Takeshima
Medicines 10 ( 7 ) 43 2023.07
Language:English Publishing type:Research paper (scientific journal)
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Total Synthesis and Monoamine Oxidase Inhibitory Activities of (±)-Entonalactam A and Its Derivatives Reviewed
Hitoshi Kamauchi, Momoka Hirata, Koichi Takao, Yoshiaki Sugita
ACS Omega 7 ( 45 ) 41804 - 41814 2022.11
Language:English Publishing type:Research paper (scientific journal)
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Antifungal activity of dehydrocurvularin for Candida spp. through the inhibition of adhesion to human adenocarcinoma cells. Reviewed
Hitoshi Kamauchi, Miho Furukawa, Yuka Kiba, Masashi Kitamura, Kanako Usui, Masanori Katakura, Koichi Takao, Yoshiaki Sugita
J. Antibiot. 75 530 - 533 2022.07
Language:English Publishing type:Research paper (scientific journal)
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Polyamines produced by an extreme thermophile are essential for cell growth at high temperature. Reviewed International journal
Akihiko Sakamoto, Masatada Tamakoshi, Toshiyuki Moriya, Tairo Oshima, Koichi Takao, Yoshiaki Sugita, Takemitsu Furuchi, Masaru Niitsu, Takeshi Uemura, Kazuei Igarashi, Keiko Kashiwagi, Yusuke Terui
J. Biochem. 172 ( 2 ) 109 - 115 2022.06
Language:English Publishing type:Research paper (scientific journal) Publisher:Oxford University Press
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A dual anti-inflammatory and anti-proliferative 3-styryl-chromone derivative sensitizes the anti-cancer effects of DNA-damaging agents on colon cancer cells by targeting HMGB1-RAGE-ERK1/2 signaling Reviewed International journal
Sei-ichi Tanuma, Takahiro Oyama, Miwa Okazawa, Hiroaki Yamazaki, Koichi Takao, Yoshiaki Sugita, Sigeru Amano, Takehiko Abe, and Hiroshi Sakagami
Int. J. Mol. Sci. 23 3426 2022.03
Language:English Publishing type:Research paper (scientific journal) Publisher:MDPI
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A benzaldehyde derivative obtained from Hypoxylon truncatum NBRC 32353 treated with hygromycin B Reviewed International journal
Hitoshi Kamauchi, Mitsuaki Suzuki, Koichi Takao, Yoshiaki Sugita
J. Antibiot. 75 ( 1 ) 1 - 8 2022.01
Language:English Publishing type:Research paper (scientific journal)
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Stimulation of the Runx2 P1 promoter by collagen-derived dipeptide prolyl-hydroxyproline bound to Foxg1 and Foxo1 in osteoblasts. Reviewed International journal
Kaho Nomura, Yoshifumi Kimira, Yoshihiro Osawa, Aya Kataoka-Matsushita, Koichi Takao, Yoshiaki Sugita, Jun Shimizu, Masahiro Wada, Hiroshi Mano
Biosci. Rep. 41 ( 12 ) BSR20210304 2021.12
Language:English Publishing type:Research paper (scientific journal) Publisher:Portland Press
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A 3-styrylchromone converted from trimebutine 3D pharmacophore possesses dual suppressive effects on RAGE and TLR4 signaling pathways. Reviewed International journal
Miwa Okazawa, Takahiro Oyama, Hideaki Abe, Hiroaki Yamazaki, Atsushi Yoshimori, Mitsutoshi Tsukimoto, Kazumi Yoshizawa, Koichi Takao, Yoshiaki Sugita, Takanori Kamiya, Fumiaki Uchiumi, Hiroshi Sakagami, Takehiko Abe, Sei-ichi Tanuma
BBRC 566 1 - 8 2021.08
Language:English Publishing type:Research paper (scientific journal)
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Synthesis and biological evaluation of 3-styrylchromone derivatives as selective monoamine oxidase B inhibitors. Reviewed International journal
Koichi Takao, Yuri Takemura, Junko Nagai, Hitoshi Kamauchi, Kaori Hoshi, Ryo Mabashi, Yoshihiro Uesawa, Yoshiaki Sugita
Bioorg. Med. Chem. 42 116255 2021.07
Authorship:Lead author Language:English Publishing type:Research paper (scientific journal)
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Synthesis and antifungal activity of polycyclic pyridone derivatives with anti-hyphal and biofilm formation activity against Candida albicans. Reviewed International journal
Hitoshi Kamauchi, Yu Kimura, Mikoto Ushiwatari, Mitsuaki Suzuki, Taishi Seki, Koichi Takao, Yoshiaki Sugita
Bioorg. Med. Chem. Lett. 37 127845 2021.04
Language:English Publishing type:Research paper (scientific journal)
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A Unique Anti-Cancer 3-Styrylchromone Suppresses Inflammatory Response via HMGB1-RAGE Signaling. Reviewed International journal
Hideaki Abe, Miwa Okazawa, Takahiro Oyama, Hiroaki Yamazaki, Atsushi Yoshimori, Takanori Kamiya, Mitsutoshi Tsukimoto, Koichi Takao, Yoshiaki Sugita, Hiroshi Sakagami, Takehiko Abe, Sei-ichi Tanuma
Medicines 8 17 2021.03
Language:English Publishing type:Research paper (scientific journal)