Papers - SUGITA Yoshiaki
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Synthesis of amide and ester derivatives of cinnamic acid and its analogs: Evaluation of their free radical scavenging and monoamine oxidase and cholinesterase inhibitory activities Reviewed
Koichi Takao, Kazuhiro Toda, Takayuki Saito, Yoshiaki Sugita
Chem. Pharm. Bull. 65 1020 - 1027 2017
Language:English Publishing type:Research paper (scientific journal)
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p-Coumaroyl malate derivatives of the Pandanus amaryllifolius leaf and their isomerization Reviewed
Ryuichiro Suzuki, Shu Kan, Yoshiaki Sugita, Yoshiaki Shirataki
Chem. Pharm. Bull. 65 1191 - 1194 2017
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure–cytotoxicity relationship of newly synthesized piperic acid esters Reviewed
10. Hiroshi Sakagami, Yoshihiro Uesawa, Yoshiko Masuda, Mineko Tomomura, Satoshi Yokose, Takaki Miyashiro, Junichi Murai, Koichi Takao, Taisei Kanamoto, Shigemi Terakubo, Hajime Kagaya, Hideki Nakashima, Yoshiaki Sugita
Anticancer Res. 37 6161 - 6168 2017
Language:English Publishing type:Research paper (scientific journal)
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Synthesis and biological evaluation of 3-benzylidene-4-chromanone derivatives as free radical scavengers and α-glucosidase inhibitors Reviewed
Koichi Takao, Marimo Yamashita, Aruki Yashiro, Yoshiaki Sugita
Chem. Pharm. Bull. 64 1203 - 1207 2016
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure–cytotoxicity relationship of 3-benzylidenechromanones Reviewed
Yoshihiro Uesawa, Hiroshi Sakagami, Hajime Kagaya, Marimo Yamashita, Koichi Takao, Yoshiaki Sugita
Anticancer Res. 36 5803 - 5812 2016
Language:English Publishing type:Research paper (scientific journal)
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2-Azolylchromone derivatives as potent and selective inhibitors of monoamine oxidases A and B Reviewed
Koichi Takao, Takayuki Saito, Daisuke Chikuda, Yoshiaki Sugita
Chem. Pharm. Bull. 64 1499 - 1504 2016
Language:English Publishing type:Research paper (scientific journal)
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Effect of spermidine analogues on cell growth of escherichia coli polyamine requiring mutant MA261 Reviewed
Taketo Yoshida, Akihiko Sakamoto, Yusuke Terui, Koichi Takao, Yoshiaki Sugita, Kaneyoshi Yamamoto, Akira Ishihama, Kazuei Igarashi, Keiko Kashiwagi
PLoS ONE 2016
Language:English Publishing type:Research paper (scientific journal)
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Synthesis and evaluation of fatty acid amides on the N-oleoylethanolamide-like activation of peroxisome proliferator activated receptor Reviewed
Koichi Takao, Kaori Noguchi, Yosuke Hashimoto, Akira Shirahata, Yoshiaki Sugita
Chem. Pharm. Bull. 63 278 - 285 2015
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure–cytotoxicity relationship of oleoylamides Reviewed
Hiroshi Sakagami, Yoshihiro Uesawa, Mariko Ishihara, Hajime Kagaya, Taisei Kanamoto, Shigemi Terakubo, Hideki Nakashima, Koichi Takao, Yoshiaki Sugita
Anticancer Res. 35 5341 - 5355 2015
Language:English Publishing type:Research paper (scientific journal)
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Effects of 3-styrylchromones on metabolic profiles and cell death in oral squamous cell carcinoma cells Reviewed
Hiroshi Sakagami, Chiyako Shimada, Yumiko Kanda, Osamu Amano, Masahiro Sugimoto, Sana Ota, Tomoyoshi Soga, Masaru Tomita, Akira Sato, Sei-ichi Tanuma, Koichi Takao and Yoshiaki Sugita
Toxicol. Rep. 2 1281 - 1290 2015
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure–cytotoxicity relationship of 3-styryl-2H-chromenes Reviewed
Yoshihiro Uesawa, Hiroshi Sakagami, Mariko Ishihara, Hajime Kagaya, Taisei Kanamoto, Shigemi Terakubo, Hideki Nakashima, Hideaki Yahagi, Koichi Takao, Yoshiaki Sugita
Anticancer Res. 35 5299 - 5308 2015
Language:English Publishing type:Research paper (scientific journal)
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Synthesis and biological evaluation of piperic acid amides as free radical scavengers and α-glucosidase inhibitors Reviewed
63 326 - 333 2015
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure-cytotoxicity relationship of 3-styrylchromones Reviewed
Chiyako Shimada, Yoshihiro Uehara, Reiko Ishii-Nozawa, Mariko Ishihara, Hajime Kagaya Taisei Kanamoto, Shigemi Terakubo, Hideki Nakashima, Koichi Takao, Yoshiaki Sugita, Hiroshi Sakagami
Anticancer Res. 34 5405 - 5412 2014
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure-cytotoxicity relationship of piperic acid amides Reviewed
Chiyako Shimada, Yoshihiro Uehara, Mariko Ishihara, Hajime Kagaya, Taisei Kanamoto, Shigemi Terakubo, Hideki Nakashima, Koichi Takao, Takaki Miyashiro, Yoshiaki Sugita, Hiroshi Sakagami
Anticancer Res. 34 4877 - 4884 2014
Language:English Publishing type:Research paper (scientific journal)
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Synthesis and biological evaluation of 3-styrylchromone derivatives as free radical scavengers and -glucosidase inhibitors Reviewed
Koichi Takao, Ryo Ishikawa, Yoshiaki Sugita
Chem. Pharm. Bull. 62 810 - 815 2014
Language:English Publishing type:Research paper (scientific journal)
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Quantitative structure-cytotoxicity relationship of phenylpropanoid amides Reviewed
Chiyako Shimada, Yoshihiro Uehara, Mariko Ishihara, Hajime Kagaya Taisei Kanamoto, Shigemi Terakubo, Hideki Nakashima, Koichi Takao, Takayuki Saito, Yoshiaki Sugita, Hiroshi Sakagami
Anticancer Res. 34 3543 - 3548 2014
Language:English Publishing type:Research paper (scientific journal)
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Development of irreversible inactivators of spermine oxidase and N1-acetylpolyamine oxidase Reviewed
Shun-suke Moriya, Toshiyuki Miura, Koichi Takao, Yoshiaki Sugita, Keijiro Samejima, Kyoko Hiramatsu, Masao Kawakita
Biol. Pharm. Bull. 37 475 - 480 2014
Language:English Publishing type:Research paper (scientific journal)
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Pentamines as substrate for human spermine oxidase Reviewed
Koichi Takao, Akira Shirahata, Keijiro Samejima, RA Casero, Kazuei Igarashi, Yoshiaki Sugita
Biol. Pharm. Bull. 36 407 - 411 2013
Language:English Publishing type:Research paper (scientific journal)
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Enhancement of gastrointestinal absorption of ovalbumin caused by spermine induces an increase in plasma histamine levels in mice sensitized to ovalbumin Reviewed
Yoshiaki Sugita, Koichi Takao, Yoshihiko, Sugino, Ryoko Kuwabara, Akira Shirahata
Biol. Pharm. Bull. 2011
Language:English Publishing type:Research paper (scientific journal)
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Assay of N1-acetylpolyamine oxidase activity with N1, N11-didansylnorspermine as the substrate by ion-pair reversed phase high performance liquid chromatography Reviewed
Koichi Takao, Yoshiaki Sugita, Akira Shirahata
Biol. Pharm. Bull. 33 ( 7 ) 1089 - 1094 2010.07
Language:English Publishing type:Research paper (scientific journal)