論文 - 杉田 義昭
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Synthesis and biological evaluation of 2-azolylmethylene-3-(2H)-benzofuranone derivatives as potent monoamine oxidases inhibitors 査読あり
Koichi Takao, Yuka Kubota, Kota Kurosaki, Hitoshi Kamauchi, Yoshihiro Uesawa, Yoshiaki Sugita
Chem. Pharm. Bull. 72 ( 1 ) 109 - 120 2024年01月
記述言語:英語
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Synthesis of 2,8-dioxabicyclo[3.3.1]nonane derivatives and their neuroprotective activities 査読あり
Hitoshi Kamauchi, Akifumi Takanashi, Mitsuaki Suzuki, Kouki Izumi, Koichi Takao, Yoshiaki Sugita
Chem. Pharm. Bull. 72 ( 1 ) 56 - 60 2024年01月
記述言語:英語
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A tricyclic aromatic polyketide isolated from the marine-derived fungus Curvularia aeria 査読あり
Hitoshi Kamauchi, Mayu Tanaka, Mitsuaki Suzuki, Miho Furukawa, Atsushi Ikeda, Chihiro Sasho, Yuka Kiba, Masashi Kitamura, Koichi Takao, Yoshiaki Sugita
Chem. Pharm. Bull. 72 ( 1 ) 98 - 101 2024年01月
記述言語:英語
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Potentiation of anticancer activity of G2/M blockers by mild hyperthermia 査読あり
Yuya Tagawa, Hiroshi Sakagami, Sei-Ichi Tamura, Shigeru Amano, Shin Uota, Kenjiro Bandow, Mineko Tomomura, Yoshihiro Uesawa, Koichi Takao, Yoshiaki Sugita, Nobuharu Yamamoto, Hideki Sakashita, Rina Nakakaji, Toshiyuki Koizumi, Kenji Mitsudo, Iwai Tohnai
Anticancer Res. 43 ( 8 ) 3429 - 3439 2023年08月
記述言語:英語
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A Comparative study of tumor-specificity and neurotoxicity between 3-styrylchromones and anti-cancer drugs 査読あり
Tomoyuki Abe, Hiroshi Sakagami, Shigeru Amano, Shin Uota, Kenjiro Bandow, Yoshihiro Uesawa, Shiori U, Hiroki Shibata, Yuri Takemura, Yu Kimura, Koichi Takao, Yoshiaki Sugita, Akira Sato, Sei-Ichi Tanuma, Hiroshi Takeshima
Medicines 10 ( 7 ) 43 2023年07月
記述言語:英語
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Total synthesis and monoamine oxidase inhibitory activities of (±)-entonalactam A and its derivertives 査読あり
Hitoshi Kamauchi, Momoka Hirata, Koichi Takao, and Yoshiaki Sugita
ACS Omega 7 41804 - 41814 2022年11月
記述言語:英語
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Antifungal activity of dehydrocurvularin for Candida spp. through the inhibition of adhesion to human adenocarcinoma cells 査読あり
Hitoshi Kamauchi , Miho Furukawa , Yuka Kiba , Masashi Kitamura , Kanako Usui , Masanori Katakura , Koichi Takao , Yoshiaki Sugita
J. Antibiot. 75 ( 9 ) 530 - 533 2022年07月
記述言語:英語
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Polyamines produced by an extreme thermophile are essential for cell growth at high temperature 査読あり
Akihiko Sakamoto, Masatada Tamakoshi, Toshiyuki Moriya, Tairo Oshima, Koichi Takao, Yoshiaki Sugita, Takemitsu Furuchi, Masaru Niitsu, Takeshi Uemura, Kazuei Igarashi, Keiko Kashiwagi, Yusuke Terui
J. Biochem. 172 ( 2 ) 109 - 115 2022年06月
記述言語:英語
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A dual anti-inflammatory and anti-proliferative 3-styryl-chromone derivative sensitizes the anti-cancer effects of DNA-damaging agents on colon cancer cells by targeting HMGB1-RAGE-ERK1/2 signaling 査読あり
Sei-ichi Tanuma, Takahiro Oyama, Miwa Okazawa, Hiroaki Yamazaki, Koichi Takao, Yoshiaki Sugita, Sigeru Amano, Takehiko Abe, and Hiroshi Sakagami
Int. J. Mol. Sci. 23 ( 7 ) 3426 2022年03月
記述言語:英語
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A benzaldehyde derivative obtained from Hypoxylon truncatum NBRC 32353 treated with hygromycin B 査読あり
Hitoshi Kamauchi, Mitsuaki Suzuki, Koichi Takao, Yoshiaki Sugita
J. Antibiot. 75 ( 1 ) 1 - 8 2022年01月
記述言語:英語
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Stimulation of the Runx2 P1 promoter by collagen-derived dipeptide prolyl-hydroxyproline bound to Foxg1 and Foxo1 in osteoblasts 査読あり
Kaho Nomura, Yoshifumi Kimira, Yoshihiro Osawa, Aya Kataoka-Matsushita, Koichi Takao, Yoshiaki Sugita, Jun Shimizu, Masahiro Wada, Hiroshi Mano
Biosci. Rep. 41 ( 12 ) 20210304 2021年12月
記述言語:英語
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A 3-styrylchromone converted from trimebutine 3D pharmacophore possesses dual suppressive effects on RAGE and TLR4 signaling pathways 査読あり
Miwa Okazawa, Takahiro Oyama, Hideaki Abe, Hiroaki Yamazaki, Atsushi Yoshimori, Mitsutoshi Tsukimoto, Kazumi Yoshizawa, Koichi Takao, Yoshiaki Sugita, Takanori Kamiya, Fumiaki Uchiumi, Hiroshi Sakagami, Takehiko Abe, Sei-ichi Tanuma
Biochem. Biophys. Res. Commun. 566 1 - 8 2021年08月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Synthesis and biological evaluation of 3-styrylchromone derivatives as selective monoamine oxidase B inhibitors 査読あり
Koichi Takao, Yuri Takemura, Junko Nagai, Hitoshi Kamauchi, Kaori Hoshi, Ryo Mabashi, Yoshihiro Uesawa, Yoshiaki Sugita
Bioorg. Med. Chem. 42 116255 2021年07月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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A Unique Anti-Cancer 3-Styrylchromone Suppresses Inflammatory Response via HMGB1-RAGE Signaling 査読あり
Hideaki Abe, Miwa Okazawa, Takahiro Oyama, Hiroaki Yamazaki, Atsushi Yoshimori, Takanori Kamiya, Mitsutoshi Tsukimoto, Koichi Takao, Yoshiaki Sugita, Hiroshi Sakagami, Takehiko Abe, Sei-ichi Tanuma
Medicines 8 17 2021年03月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Synthesis and antifungal activity of polycyclic pyridone derivatives with anti-hyphal and biofilm formation activity against Candida albicans 査読あり
Hitoshi Kamauchi, Yu Kimura, Mikoto Ushiwatari, Mitsuaki Suzuki, Taishi Seki, Koichi Takao, Yoshiaki Sugita
Bioorg. Med. Chem. Lett. 37 127845 2021年02月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Syntheses and evaluation of 2- or 3-(N-cyclicamino)chromone derivatives as monoamine oxidase inhibitors 査読あり
Koichi Takao, Tsukasa Sakatsume, Hitoshi Kamauchi and Yoshiaki Sugita
Chem. Pharm. Bull. 68 ( 11 ) 1082 - 1089 2020年11月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Quantification of the ability of natural products to prevent herpes virus infection 査読あり
Kunihiko Fukuchi, Hiroshi Sakagami, Yoshiaki Sugita, Koichi Takao, Daisuke Asai, Shigemi Terakubo, Hiromu Takemura, Hirokazu Ohno, Misaki Horiuchi, Madoka Suguro, Tomohiro Fujisawa, Kazuki Toeda, Hiroshi Oizumi, Toshikazu Yasui, Takaaki Oizumi
Medicines (MDPI) 7 ( 10 ) 64 2020年10月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Syntheses and crystal structures of two piperine derivatives 査読あり
Toshinari Ezawa, Yutaka Inoue, Isamu Murata, Mitsuaki Suzuki, Koichi Takao, Yoshiaki Sugita, Ikuo Kanamoto
Acta Crystallogr. E. Crystallogr. Commun. 76 ( 5 ) 646 - 650 2020年05月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Further quantitative structure–cytotoxicity relationship analysis of 3-styrylchromones 査読あり
Koichi Takao, Kaori Hoshi, Hiroshi Sakagami, Haixia Shi, Kenjiro Bandow, Junko Nagai, Yoshihiro Uesawa, Akito Tomomura, Mineko Tomomura, Yoshiaki Sugita
Anticancer Res. 40 ( 1 ) 87 - 95 2020年01月
記述言語:英語 掲載種別:研究論文(学術雑誌)
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Synthesis and pharmacological evaluation of childinin E and several derivatives as anti-hyphal formation inhibitors against Candida albicans 査読あり
Hitoshi Kamauchi Momoka Hirata, Koichi Takao, Yoshiaki Sugita
Tetrahedron Lett. 61 ( 49 ) 152588 2020年
記述言語:英語 掲載種別:研究論文(学術雑誌)